Aromatase Inhibitor
FOR HARDCORE USERS ONLY
ErgoPharm decided to come up with 6-OXO Extreme for a couple of very good reasons. ErgoPharm felt that many of our customers desired an even more potent t-boost than 6-OXO provided, and they had the technology to deliver the product. So they made it. They did not just throw this formula together however. They undertook the due testing to prove to themselves that this product had the ability to stimulate t- levels beyond even the range of upper normal - indeed it stimulates levels well into the supraphysiological range.
6-OXO Extreme begins of course with the time tested natural metabolite 4-etioallocholen-3,6,17-trione. As you already know, this compound acts in the body as an inhibitor of the enzyme aromatase, which governs the production of estrogen hormones in the body. By reducing the levels of estrogen in the body a compensatory reaction in the brain is initiated leading to an increase in the secretion of LH which in turn causes testosterone production to increase.
To complement the anti-aromatase action of 6-OXO they added a natural ingredient that acts as an estrogen receptor antagonist (ERA). An ERA is a compound that binds to estrogen receptors and blocks them from interacting with circulating estrogen hormones. However, unlike regular estrogen hormones the ERA does not result in a subsequent activation of the estrogen "signal", the action that is supposed to happen when a hormone binds to its receptor. The ERA therefore prevents the circulating estrogens in your body from having a chance to do their thing.
The ERA ErgoPharm chose is perhaps the single most amazing natural compound they have ever come across. It is called resveratrol and it is found in red wine. You may have heard of resveratrol as it has gotten alot of media attention lately due to recent research showing it to have amazing life extension and anti-aging properties. But what the media has not mentioned, and the researchers have not seemingly recognized, is that resveratrol intake has the ability to raise testosterone levels in males.
Resveratrol has a problem though, and it concerns its bioavailability. When you consume resveratrol it is absorbed adequately into the blood stream but after that it is very quickly sulfated and glucuronidated by enzymes. What this means is that it is transformed into inactive derivatives meant for elimination from the body. To get an active quantity of resveratrol into the body you have to overcome this problem. This is done by simultaneously ingesting compounds (quercetin and piperine) that will use up these enzymes preferentially, leaving the resveratrol free to circulate in the body. A large dose must also be taken, as the enzyme blocking will only be partially effective.
So with effective aromatase inhibition plus estrogen receptor blockade we have a two pronged attack on estrogen mediated HPTA feedback inhibition. With added ZMA to address any possible interfering mineral deficiencies, this formula will produce extraordinary results - better than anything presently on the market by far!!
Suggested Use: As a dietary supplement, take 1-2 servings per day with food. Take for cycles of 4 to 8 weeks.
Also Available: 6-OXO & 11-OXO
